Synthesis of 1,2,4-triazoles employing isocyanides

Design, Synthesis, and Antifouling Activity of Glucosamine-Based Isocyanides

Biofouling, an undesirable accumulation of organisms on sea-immersed structures such as ship hulls and fishing nets, is a serious economic issue whose effects include oil wastage and clogged nets. Organotin compounds were utilized since the 1960s as an antifouling material; however, the use of such compounds was later banned by the International Maritime Organization (IMO) due to their high tox...

Synthesis of Copolymers of Isocyanides Derived from Alanylserine and Alanylhistidine1

Synthesis and Microwave Spectroscopic Study of Fluorinated Methyl Isocyanides

für Naturforschung in cooperation with the Max Planck Society for the Advancement of Science under a Creative Commons Attribution 4.0 International License. Dieses Werk wurde im Jahr 2013 vom Verlag Zeitschrift für Naturforschung in Zusammenarbeit mit der Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. digitalisiert und unter folgender Lizenz veröffentlicht: Creative Commons Namen...

Synthesis of Antimicrobial N-Phthaloyl-alanyl-derived Amidophosphates and Triazoles

N-Phthaloyl-alanylazide reacts smoothly with trialkyl phosphites producing the corresponding αaminophosphates. With dialkyl hydrogenphosphonates in the presence of benzoyl peroxide, amidophosphates were the isolated products whereas the oxoaziridin-1-yl-phosphonic diamide was preferentially provided from the reaction of the azide with tris(dimethylamino)phosphine. The azide was also allowed to ...

"Flash" solvent-free synthesis of triazoles using a supported catalyst.

A solvent-free synthesis of 1,4-disubstituted-1,2,3-triazoles using neat azides and alkynes and a copper(I) polymer supported catalyst (Amberlyst) A21*CuI) is presented herein. As it provides the products in high yields and purities within minutes, this method thus being characterized as a "flash" synthesis, and was exemplified through the synthesis of a 24-compound library on a small scale.